Home GPCR & G Protein S1P Receptor S1PR1 Agonists

S1PR1 Agonists

  • S1PR1
  • S1PR4
  • S1PR5
  • SphK
N. Cat. Nome del prodotto Informazioni Selettivo / Pan IC50 / Ki
S7179 BAF312 (Siponimod) BAF312 (Siponimod) is a next-generation S1P receptor modulator, selective for S1P1 and S1P5 receptors with EC50 of 0.39 nM and 0.98 nM, exhibits >1000-fold selectivity over S1P2, S1P3 and S1P4 receptors. Phase 3. Pan S1P1 receptor, EC50: 0.39 nM