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NMDA receptor-Selettivo Antagonists

  • NMDA receptor
  • AMPA receptor
  • mGluR2
  • mGluR3
  • mGluR4
  • mGluR5
N. Cat. Nome del prodotto Informazioni Selettivo / Pan IC50 / Ki
S2857 MK-801 (Dizocilpine) MK-801 (Dizocilpine) is a potent N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 30.5 nM. Selective NMDA Receptor, Ki: 30.5 nM
S2876 (-)-MK 801 Maleate MK-801 is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes. Selective NMDA Receptor, Kd: 37.2 nM
S4091 Ifenprodil Tartrate Ifenprodil is an atypical noncompetitive antagonist at the NMDA receptor, it interacts with high affinity at a homogeneous population of NMDA receptors in neonatal rat forebrain with IC50 of 0.3 μM. Selective NMDA Receptor, IC50: 0.3 μM
S7072 NMDA (N-Methyl-D-aspartic acid) NMDA（N-Methyl-D-aspartic acid）is a specific agonist for NMDA receptor mimicking the action of glutamate, the neurotransmitter which normally acts at that receptor. Phase 4. Selective
S1614 Riluzole Riluzole is a drug used to treat amyotrophic lateral sclerosis. Selective