D5 receptor Antagonists

  • D1 receptor
  • D2 receptor
  • D3 receptor
  • D5 receptor
  • DAT
  • D4 receptor
N. Cat. Nome del prodotto Informazioni Selettivo / Pan IC50 / Ki
S1771 Chlorprothixene Chlorprothixene has strong binding affinities to dopamine and histamine receptors, such as D1, D2, D3, D5, H1, 5-HT2, 5-HT6 and 5-HT7, with Ki of 18 nM, 2.96 nM, 4.56 nM, 9 nM, 3.75 nM, 9.4 nM, 3 nM and 5.6 nM, respectively. Pan D5 receptor, Ki: 9 nM