D4 receptor Agonists | Antagonists

  • D1 receptor
  • D2 receptor
  • D3 receptor
  • D5 receptor
  • DAT
  • D4 receptor
N. Cat. Nome del prodotto Informazioni Selettivo / Pan IC50 / Ki
S2011 Pramipexole 2HCl Monohydrate Pramipexole 2HCl Monohydrate is a partial/full D2S, D2L, D3, D4, receptor agonist with a Ki of 3.9, 2.2, 0.5, 5.1 nM. Pan D4 receptor, Ki: 5.1 nM
S2460 Pramipexole Pramipexole is a partial/full D2S, D2L, D3, D4 receptor agonist with a Ki of 3.9, 2.2, 0.5 and 5.1 nM for D2S, D2L, D3, D4 receptor, respectively. Pan D4 receptor, Ki: 5.1 nM
S4086 Loxapine Succinate Loxapine Succinate is a D2DR and D4DR inhibitor, serotonergic receptor antagonist and also a dibenzoxazepine anti-psychotic agent. Pan D4 receptor (human), Ki: 7.5 nM