Home Neuronal Signaling -GPCR & G Protein Dopamine Receptor D3 receptor-Selettivo Agonists | Antagonists

D3 receptor-Selettivo Agonists | Antagonists

  • D1 receptor
  • D2 receptor
  • D3 receptor
  • D5 receptor
  • DAT
  • D4 receptor
N. Cat. Nome del prodotto Informazioni Selettivo / Pan IC50 / Ki
S2168 PD128907 HCl PD 128907 HCl is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor. Selective D3 receptor, EC50: 0.64 nM
S2460 Pramipexole Pramipexole is a partial/full D2S, D2L, D3, D4 receptor agonist with a Ki of 3.9, 2.2, 0.5 and 5.1 nM for D2S, D2L, D3, D4 receptor, respectively. Pan D3 receptor, Ki: 0.5 nM
S2011 Pramipexole 2HCl Monohydrate Pramipexole 2HCl Monohydrate is a partial/full D2S, D2L, D3, D4, receptor agonist with a Ki of 3.9, 2.2, 0.5, 5.1 nM. Pan D3 receptor, Ki: 0.5 nM
S1771 Chlorprothixene Chlorprothixene has strong binding affinities to dopamine and histamine receptors, such as D1, D2, D3, D5, H1, 5-HT2, 5-HT6 and 5-HT7, with Ki of 18 nM, 2.96 nM, 4.56 nM, 9 nM, 3.75 nM, 9.4 nM, 3 nM and 5.6 nM, respectively. Pan D3 receptor, Ki: 4.56 nM
S2437 Rotundine Rotundine (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM. Pan D3 receptor, IC50: 3.25 μM